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Attributs	Valeurs
type	work Issue
Is Part Of	http://hub.abes.fr/acs/periodical/jmcmar/1989/volume_32
has manifestation of work	http://hub.abes.fr/acs/periodical/jmcmar/1989/volume_32/issue_4/m/print http://hub.abes.fr/acs/periodical/jmcmar/1989/volume_32/issue_4/m/web
issue	4
is Is Part Of of	Hybrid cholecystokinin (CCK) antagonists: new implications in the design and modification of CCK antagonists Topography and conformational preferences of 6,7,8,9-tetrahydro-1-hydroxy-N,N-dipropyl-5H-benzocyclohepten-6-ylamine. A rationale for the dopaminergic inactivity Book Reviews Analogs of cisplatin derived from diaminodideoxytetritols. Synthesis and activity against the ADJ/PC6 plasmacytoma in mice A minor modification of residue 1 in potent vasopressin antagonists dramatically reduces agonist activity Benzofurans as mechanism-based inhibitors of dopamine .beta.-hydroxylase Synthesis, DNA-binding properties, and antitumor activity of novel distamycin derivatives Approaches to isozyme-specific inhibitors. 16. A novel methyl-C5' covalent adduct of L-ethionine and .beta.,.gamma.-imido-ATP as a potent multisubstrate inhibitor of rat methionine adenosyltransferases Masthead Hydroxyacetophenone-derived antagonists of the peptidoleukotrienes New sensitizers for photodynamic therapy. Controlled synthesis of purpurins and their effect on normal tissue Synthesis and biological evaluation of de(acetylglucosaminyl)didehydrodeoxy derivatives of teicoplanin antibiotics 2'-Fluorinated isonucleosides. 1. Synthesis and biological activity of some methyl 2'-deoxy-2'-fluoro-2'-pyrimidinyl-D-arabinopyranosides Identification of structural requirements for analogs of atrial natriuretic peptide (ANP) to discriminate between ANP receptor subtypes Topographic probes of angiotensin and receptor: potent angiotensin II agonist containing diphenylalanine and long-acting antagonists containing biphenylalanine and 2-indan amino acid in position 8 Carboxyalkyl dipeptides with atrial natriuretic factor potentiating and antihypertensive activity Synthesis and pharmacology of a series of 3- and 4-(phosphonoalkyl)pyridine- and -piperidine-2-carboxylic acids. Potent N-methyl-D-aspartate receptor antagonists Synthesis and D2 dopaminergic activity of pyrrolidinium, tetrahydrothiophenium, and tetrahydrothiophene analogs of sulpiride Synthesis of congeners and prodrugs. 3. Water-soluble prodrugs of taxol with potent antitumor activity Design and synthesis of propranolol analogs as serotonergic agents Computer assisted design and synthesis of novel aldose reductase inhibitors Retinobenzoic acids. 2. Structure-activity relationships of chalcone-4-carboxylic acids and flavone-4'-carboxylic acids Quinazoline antifolates inhibiting thymidylate synthase: 2-desamino derivatives with enhanced solubility and potency Comparison of the biological effects of selected 5,8-dideazafolate analogs with their 2-desamino counterparts Analysis of the in vitro antiviral activity of certain ribonucleosides against parainfluenza virus using a novel computer aided receptor modeling procedure Synthesis of some novel potent and selective catechol O-methyltransferase inhibitors Conformationally restricted analogs of the muscarinic agent N-methyl-N-(1-methyl-4-pyrrolidino-2-butynyl)acetamide Resolved N,N-dialkylated 2-amino-8-hydroxytetralins: stereoselective interactions with 5-HT1A receptors in the brain [(1H-Imidazol-1-yl)methyl]- and [(3-pyridinyl)methyl]pyrroles as thromboxane synthetase inhibitors Potential antitumor agents. 58. Synthesis and structure-activity relationships of substituted xanthenone-4-acetic acids active against the colon 38 tumor in vivo Synthesis and evaluation of the pharmacological activity of rigid analogs of sympathomimetic catecholamines derived from bicyclo[2.2.1]heptane

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