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Attributs	Valeurs
type	work Issue
Is Part Of	http://hub.abes.fr/acs/periodical/jmcmar/2003/volume_46
has manifestation of work	http://hub.abes.fr/acs/periodical/jmcmar/2003/volume_46/issue_14/m/print http://hub.abes.fr/acs/periodical/jmcmar/2003/volume_46/issue_14/m/web
Date Copyrighted	2003
Rights	Copyright © 2003 American Chemical Society
issue	14
Rights Holder	American Chemical Society
is Is Part Of of	Synthesis of 1-Boraadamantaneamine Derivatives with Selective Astrocyte vsC6 Glioma Antiproliferative Activity. A Novel Class of Anti-Hepatitis C Agentswith Potential to Bind CD81 A Convergent Approach to Cryptophycin 52 Analogues: Synthesis andBiological Evaluation of a Novel Series of Fragment A Epoxides andChlorohydrins A Quantitative Structure−Activity Relationship and Pharmacophore ModelingInvestigation of Aryl-X and Heterocyclic Bisphosphonates as Bone ResorptionAgents Development of Natural Product-Derived Receptor Tyrosine Kinase InhibitorsBased on Conservation of Protein Domain Fold Design and Synthesis of Poly ADP-ribose Polymerase-1 Inhibitors. 2. BiologicalEvaluation of Aza-5[H]-phenanthridin-6-ones as Potent, Aqueous-SolubleCompounds for the Treatment of Ischemic Injuries New Pyrimido[5,4-b]indoles as Ligands for α1-Adrenoceptor Subtypes Novel Selective Hindlimb Vasodilators: Synthesis and Biological Activity of1-Acyl-4-aminopiperidine Derivatives N-(3-Acyloxy-2-benzylpropyl)-N‘-[4-(methylsulfonylamino)benzyl]thioureaAnalogues: Novel Potent and High Affinity Antagonists and Partial Antagonistsof the Vanilloid Receptor Higher-End Serotonin Receptors: 5-HT5, 5-HT6, and 5-HT7 Modern Methods of Drug Discovery Edited byAlexander Hillisch and Rolf Hilgenfeld. BirkhäuserVerlag, Basel, Switzerland. viii + 292 pp. 17 × 24 cm.ISBN 3-7643-6081-X. 127.00 euro. Dual Protein Farnesyltransferase−Geranylgeranyltransferase-I Inhibitors asPotential Cancer Chemotherapeutic Agents Nuclear Hormone Receptor Targeted Virtual Screening Design and Synthesis of 4,6-Di-tert-butyl-2,3-dihydro-5-benzofuranols as a NovelSeries of Antiatherogenic Antioxidants Docking and Database Screening Reveal New Classes of Plasmodiumfalciparum Dihydrofolate Reductase Inhibitors Estrogen Receptor Modulators: Identification and Structure−ActivityRelationships of Potent ERα-Selective Tetrahydroisoquinoline Ligands Identification of (3R)-7-Hydroxy-N-((1S)-1-{[(3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethyl-1-piperidinyl]methyl}-2-methylpropyl)-1,2,3,4-tetrahydro-3-isoquinolinecarboxamide as a Novel Potent and Selective Opioid κ ReceptorAntagonist Novel Potent 5-HT1F Receptor Agonists: Structure−Activity Studies of a Seriesof SubstitutedN-[3-(1-Methyl-4-piperidinyl)-1H-pyrrolo[3,2-b]pyridin-5-yl]amides Carbon Isosteres of the 4-Aminopyridine Substructure of Chloroquine: Effectson pKa, Hematin Binding, Inhibition of Hemozoin Formation, and ParasiteGrowth Histamine-Releasing Activity and Binding to the FcεRIα Human Mast CellReceptor Subunit of Mast Cell Degranulating Peptide Analogues with AlanineSubstitutions A Selective Human H4-Receptor Agonist: (−)-2-Cyano-1-methyl-3-{(2R,5R)-5-[1H-imidazol-4(5)-yl]tetrahydrofuran-2-yl}methylguanidine Novel DualInhibitors of AChE and MAO Derived from HydroxyAminoindan and Phenethylamine as Potential Treatment for Alzheimer's Disease. Simplified Discodermolide Analogues: Synthesis and Biological Evaluation of4-epi-7-Dehydroxy-14,16-didemethyl-(+)-discodermolides asMicrotubule-Stabilizing Agents 4-Aryl-3-(hydroxyalkyl)quinolin-2-ones: Novel Maxi-K Channel OpeningRelaxants of Corporal Smooth MuscleTargeted for Erectile Dysfunction Bioactive Peptidic Analogues and Cyclostereoisomers of the MinimalAntinociceptive Histogranin Fragment-(7−10) Design, Synthesis, and Evaluation of Psorospermin/Quinobenzoxazine Hybridsas Structurally Novel Antitumor Agents A New Biotin Derivative−DOTA Conjugate as a Candidate for PretargetedDiagnosis and Therapy of Tumors Opioid Binding and in Vitro Profiles of a Series of4-Hydroxy-3-methoxyindolomorphinans. Transformation of a δ-Selective Ligandinto a High Affinity κ-Selective Ligand by Introduction of a 5,14-SubstitutedBridge Development and Validation of k-Nearest-Neighbor QSPR Models of MetabolicStability of Drug Candidates Information Decay in Molecular Docking Screens against Holo, Apo, andModeled Conformations of Enzymes Synthesis and Evaluation of 17α-20E-21-(4-Substitutedphenyl)-19-norpregna-1,3,5(10),20-tetraene-3,17β-diols as Probes for the EstrogenReceptor α Hormone Binding Domain Studies on the Synthesis and Biological Properties of Non-Carrier-Added[125I and 131I]-Labeled Arylalkylidenebisphosphonates: Potent Bone-Seekers forDiagnosis and Therapy of Malignant Osseous Lesions Structure−Activity Relationship Comparison of (S)-2β-Substituted3α-(Bis[4-fluorophenyl]methoxy)tropanes and (R)-2β-Substituted3β-(3,4-Dichlorophenyl)tropanes at the Dopamine Transporter Structure−Activity Relationships and Mechanism of Action of AntitumorBenzo[b]pyrano[3,2-h]acridin-7-one Acronycine Analogues Synthesis and Anticonvulsant Activity of Novel Bicyclic Acidic Amino Acids Design, Synthesis, and Biological Properties of NewBis(acridine-4-carboxamides) as Anticancer Agents Structural Determinants of Selective Thyromimetics Cardiovascular Pharmacotherapeutics. SecondEdition Edited by William H. Frishman, Edmund H.Sonnenblick, and Domenic A. Sica. McGraw-Hill Medical Publishing Division, New York. 2003. xxiv + 1072pp. 22.5 × 29 cm. ISBN 0-07-136981-3. $159.00. Design, Synthesis, and Evaluation ofNovel Boronic-Chalcone Derivatives asAntitumor Agents Dihydrofolate Reductase Mutant withExceptional Resistance to Methotrexatebut Not to Trimetrexate

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