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Attributs	Valeurs
type	work Issue
Is Part Of	http://hub.abes.fr/acs/periodical/jmcmar/2006/volume_49
has manifestation of work	http://hub.abes.fr/acs/periodical/jmcmar/2006/volume_49/issue_24/m/print http://hub.abes.fr/acs/periodical/jmcmar/2006/volume_49/issue_24/m/web
Date Copyrighted	2006
Rights	Copyright © 2006 American Chemical Society
issue	24
Rights Holder	American Chemical Society
is Is Part Of of	QSAR Modeling of Human Serum Protein Binding with Several Modeling Techniques UtilizingStructure−Information Representation Tricyclic Imidazoline Derivatives as Potent and Selective Adenosine A1 Receptor Antagonists Potent, Selective, and Orally Efficacious Antagonists of Melanin-Concentrating HormoneReceptor 1 Discovery of a New Class of Macrocyclic Antagonists to the Human Motilin Receptor Synthesis and Biological Evaluation of New Asymmetrical Bisintercalators as PotentialAntitumor Drugs Carbonic Anhydrase Inhibitors: Clash with Ala65 as a Means for Designing Inhibitors withLow Affinity for the Ubiquitous Isozyme II, Exemplified by the Crystal Structure of theTopiramate Sulfamide Analogue Discovery of Conformationally ConstrainedTetracyclic Compounds as Potent Hepatitis CVirus NS5B RNA Polymerase Inhibitors Pyrrolo[1,2-b][1,2,5]benzothiadiazepines (PBTDs): A New Class of Agentswith High Apoptotic Activity in Chronic Myelogenous Leukemia K562 Cells and in Cells from Patients at Onset and WhoWere Imatinib-Resistant. New Orally Active Derivatives of Artemisinin with High Efficacy against Multidrug-ResistantMalaria in Mice Potent and Orally Bioavailable 8-Bicyclo[2.2.2]octylxanthines as Adenosine A1 ReceptorAntagonists Conjugation of Adenosine and Hexa-(d-arginine) Leads to a Nanomolar Bisubstrate-AnalogInhibitor of Basophilic Protein Kinases Novel Schiff Base Copper Complexes of Quinoline-2 Carboxaldehyde as Proteasome Inhibitorsin Human Prostate Cancer Cells Application of Phosphoramidate ProTide Technology Significantly Improves Antiviral Potencyof Carbocyclic Adenosine Derivatives WB4101-Related Compounds: New, Subtype-Selective α1-Adrenoreceptor Antagonists (orInverse Agonists?) Synthesis and Radioligand Binding Studies of Methoxylated 1,2,3,4-TetrahydroisoquinoliniumDerivatives as Ligands of the Apamin-Sensitive Ca2+-Activated K+ Channels Design and Synthesis of NovelIsoquinoline-3-nitriles as Orally BioavailableKv1.5 Antagonists for the Treatment ofAtrial Fibrillation Discovery and Development of 5-[(5S,9R)-9-(4-Cyanophenyl)-3-(3,5-dichlorophenyl)-1-methyl-2,4-dioxo-1,3,7-triazaspiro[4.4]non-7-yl-methyl]-3-thiophenecarboxylic Acid(BMS-587101)A Small Molecule Antagonist ofLeukocyte Function Associated Antigen-1 Design, Synthesis, and Preliminary Evaluation of Doxazolidine Carbamates as ProdrugsActivated by Carboxylesterases Selective Angiotensin II AT2 Receptor Agonists: Arylbenzylimidazole Structure−ActivityRelationships 1,4,5,6-Tetrahydropyrrolo[3,4-c]pyrazoles: Identification of a Potent Aurora Kinase Inhibitorwith a Favorable Antitumor Kinase Inhibition Profile MacrocyclicInhibitors of β-Secretase: Functional Activity in an AnimalModel. Estimation of Volume of Distribution in Humans from High Throughput HPLC-BasedMeasurements of Human Serum Albumin Binding and Immobilized Artificial MembranePartitioning Discovering Inhibitors of Human Sirtuin Type 2: Novel Structural Scaffolds Analysis of the Structure−Activity Relationship of Four Herpesviral UL97 Subfamily ProteinKinases Reveals Partial but not Full Functional Conservation† Further Synthetic and Biological Studies on Vitamin D Hormone Antagonists Based onC24-Alkylation and C2α-Functionalization of 25-Dehydro-1α-hydroxyvitamin D3-26,23-lactones 6-(4-Chlorophenyl)-3-substituted-thieno[3,2-d]pyrimidin-4(3H)-one-BasedMelanin-Concentrating Hormone Receptor 1 Antagonist Synthesis of DNA-Directed Pyrrolidinyl and Piperidinyl Confined AlkylatingChloroalkylaminoanthraquinones: Potential for Development of Tumor-Selective N-Oxides The Design, Synthesis, and Evaluation of Organ-Specific Iron Chelators Endoperoxide Derivatives from Marine Organisms: 1,2-Dioxanes of the Plakortin Family asNovel Antimalarial Agents A 2.13 Å Structure of E. coli Dihydrofolate Reductase Bound to a Novel Competitive InhibitorReveals a New Binding Surface Involving the M20 Loop Region Acyl Glucuronides: Biological Activity, Chemical Reactivity, and Chemical Synthesis Solution Structure of Mouse Cripto CFC Domain and Its Inactive Variant Trp107Ala Synthesis andProperties of Benzo[a]phenoxazinium Chalcogen Analogues asNovel Broad-Spectrum Antimicrobial Photosensitizers. Structure−Activity Relationships of a Novel Series of Urotensin II Analogues: Identification ofa Urotensin II Antagonist Synthetic Inhibitors of Cytochrome P-450 2A6: Inhibitory Activity, Difference Spectra,Mechanism of Inhibition, and Protein Cocrystallization Substituted trans-Stilbenes, Including Analogues of the Natural Product Resveratrol, Inhibit theHuman Tumor Necrosis Factor Alpha-Induced Activation of Transcription Factor NuclearFactor KappaB Fragment-Based Drug Design: How Big Is Too Big? Synthesis and Structure−Activity Relationships of Uracil Nucleotide Derivatives and Analoguesas Agonists at Human P2Y2, P2Y4, and P2Y6 Receptors

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