Abstract
| - Dichloroacetamides, on heating with benzotriazole, morpholine, and triethylamine, produce, in a one-potreaction, α-benzotriazolyl-α-morpholinoacetamides 4a,b. Intermediates 4a and 4b react with nucleophiles such asallylsilanes, silyl ethers, and organozinc reagents to afforddiverse α-morpholinoamides.
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