Abstract
| - Enantiopure 2-(tributylstannyl)pyrrolidine hydroiodide maybe prepared in excellent yield by TMSI treatment of thecorresponding N-Boc compound, which is in turn preparedby asymmetric deprotonation (s-BuLi·sparteine) and stannylation, as described in the literature. Crystals of thehydroiodide salt suitable for X-ray analysis were obtained,and although there is some disorder about the butyl groups,analysis using anomalous dispersion establishes the absoluteconfiguration as S.
|