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Attributs	Valeurs
type	work Issue
Is Part Of	http://hub.abes.fr/acs/periodical/jmcmar/2005/volume_48
has manifestation of work	http://hub.abes.fr/acs/periodical/jmcmar/2005/volume_48/issue_9/m/print http://hub.abes.fr/acs/periodical/jmcmar/2005/volume_48/issue_9/m/web
Date Copyrighted	2005
Rights	Copyright © 2005 American Chemical Society
issue	9
Rights Holder	American Chemical Society
is Is Part Of of	Antitumor Effects of Two Novel Naturally Occurring Terpene QuinonesIsolated from the Mediterranean Ascidian Aplidium conicum HierS: Hierarchical Scaffold Clustering Using Topological Chemical Graphs Conformation Mining: An Algorithm for Finding Biologically RelevantConformations Platinum(II) Complexes with Antitumoral/Antiviral Aromatic Heterocycles: Effect of Glutathione upon in Vitro Cell Growth Inhibition Synthesis and Antibacterial Activity of the 4-Quinolone-3-carboxylic AcidDerivatives Having a Trifluoromethyl Group as a Novel N-1 Substituent Successful in Silico Discovery of Novel Nonsteroidal Ligands for Human SexHormone Binding Globulin Molecular Dynamics Simulation of the Ligand Binding Domain of Farnesoid XReceptor. Insights into Helix-12 Stability and Coactivator Peptide Stabilizationin Response to Agonist Binding A Bioavailability Score Frontal Affinity Chromatography with MS Detection of EphB2 Tyrosine KinaseReceptor. 2. Identification of Small-Molecule Inhibitors via Coupling withVirtual Screening Synthesis and Biological Evaluation of 14-Alkoxymorphinans. 22. Influence ofthe 14-Alkoxy Group and the Substitution in Position 5 in14-Alkoxymorphinan-6-ones on in Vitro and in Vivo Activities C-5-Disubstituted Barbiturates as Potential Molecular Probes for NoninvasiveMatrix Metalloproteinase Imaging Structure−Activity Relationships of Fluorinated Lysophosphatidic AcidAnalogues DASH: A Novel Analysis Method for Molecular Dynamics Simulation Data.Analysis of Ligands of PPAR-γ Convergent Synthesis and Pharmacology of SubstitutedTetrazolyl-2-amino-3-(3-hydroxy-5-methyl-4-isoxazolyl)propionic acid Analogues Synthesis and Antibacterial Activity of1-(2-Fluorovinyl)-7-substituted-4-quinolone-3-carboxylic Acid Derivatives,Conformationally Restricted Analogues of Fleroxacin On the Binding of Indeno[1,2-c]isoquinolines in the DNA−Topoisomerase ICleavage Complex Design of Benzophenone-Containing Photoactivatable Linear VasopressinAntagonists: Pharmacological and Photoreactive Properties Adenosine Kinase Inhibitors. 4. 6,8-Disubstituted Purine NucleosideDerivatives. Synthesis, Conformation, and Enzyme Inhibition Synthesis and Cytotoxic Evaluation of Combretafurazans http://hub.abes.fr/acs/periodical/jmcmar/2005/volume_48/issue_9/101021jm058193u/w Symmetrical Bis-Quinolinium Compounds: New Human Choline KinaseInhibitors with Antiproliferative Activity against the HT-29 Cell Line Ligand-Based Prediction of Active Conformation by 3D-QSAR FlexibilityDescriptors and Their Application in 3+3D-QSAR Models Structural Requirements for Factor Xa Inhibition by 3-Oxybenzamides withNeutral P1 Substituents: Combining X-ray Crystallography, 3D-QSAR, andTailored Scoring Functions New Drug Approval Process. Accelerating GlobalRegistrations. 4th Edition Edited by Richard A.Guarino. Marcel Dekker, New York. 2004. xiv + 635 pp.16 × 23.5 cm. ISBN 0824750411. $164.00. Thermodynamic Analysis of Interactionsbetween N-Linked Sugar Chains andF-Box Protein Fbs1 Calculating Virtual log P in the Alkane/Water System (log PNalk) and Its DerivedParameters Δlog PNoct-alk and log DpHalk Computational Strategies in Discovering Novel Non-nucleoside Inhibitors ofHIV-1 RT Thyroid Receptor Ligands. 3. Design andSynthesis of3,5-Dihalo-4-alkoxyphenylalkanoic Acidsas Indirect Antagonists of the ThyroidHormone Receptor Bisphosphonate Inhibitors of Toxoplasma gondi Growth: In Vitro, QSAR, andIn Vivo Investigations Identification and Structure−ActivityRelationship of Phenolic AcylHydrazones as Selective Agonists for theEstrogen-Related Orphan NuclearReceptors ERRβ and ERRγ Enantiomerically Pure Hexahydropyrazinoquinolines as Potent and SelectiveDopamine 3 Subtype Receptor Ligands Synthesis and Biological Evaluation ofAminopolyamines Discovery of Diphenyloxazole andNδ-Z-Ornithine Derivatives as HighlyPotent and Selective HumanProstaglandin EP4 Receptor Antagonists 1,5-Diarylpyrrole-3-acetic Acids and Esters as Novel Classes of Potent andHighly Selective Cyclooxygenase-2 Inhibitors Identification of Novel Low Molecular Weight CXCR4 Antagonists by StructuralTuning of Cyclic Tetrapeptide Scaffolds 1-(5-Chloro-2-alkoxyphenyl)-3-(5-cyano-pyrazi-2-yl)ureas as Potent and SelectiveInhibitors of Chk1 Kinase: Synthesis,Preliminary SAR, and BiologicalActivities N-Terminal Fatty Acylated His-dPhe-Arg-Trp-NH2 Tetrapeptides: Influence ofFatty Acid Chain Length on Potency and Selectivity at the Mouse MelanocortinReceptors and Human Melanocytes “In Situ Cross-Docking” ToSimultaneously Address Multiple Targets Synthesis and Pharmacology of 6-Substituted Benztropines: Discovery of NovelDopamine Uptake Inhibitors Possessing Low Binding Affinity to the DopamineTransporter Synthesis and in Vitro and in Vivo Antitumor Activity of2-Phenylpyrroloquinolin-4-ones Discovery of a β-MSH-Derived MC-4RSelective Agonist Morphiceptin Analogues Containing a Dipeptide Mimetic Structure: AnInvestigation on the Bioactive Topology at the μ-Receptor Toward a Novel Class of AntithromboticCompounds with Dual Function.Discovery of 1,4-Benzoxazin-3(4H)-oneDerivatives Possessing ThrombinInhibitory and Fibrinogen ReceptorAntagonistic Activities Class II (IIa)-Selective Histone Deacetylase Inhibitors. 1. Synthesis andBiological Evaluation of Novel (Aryloxopropenyl)pyrrolyl Hydroxyamides Discovery of 3-[(4,5,7-Trifluorobenzothiazol-2-yl)methyl]indole-N-acetic Acid(Lidorestat) and Congeners as Highly Potent and Selective Inhibitors of AldoseReductase for Treatment of Chronic Diabetic Complications

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