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Attributs	Valeurs
type	work Issue
Is Part Of	http://hub.abes.fr/acs/periodical/jmcmar/2005/volume_48
has manifestation of work	http://hub.abes.fr/acs/periodical/jmcmar/2005/volume_48/issue_23/m/print http://hub.abes.fr/acs/periodical/jmcmar/2005/volume_48/issue_23/m/web
Date Copyrighted	2005
Rights	Copyright © 2005 American Chemical Society
issue	23
Rights Holder	American Chemical Society
is Is Part Of of	Design, Synthesis, and Binding Studies of New Potent Ligands of CannabinoidReceptors Novel Benzopyridothiadiazepines as Potential Active Antitumor Agents Enantioselective Nonsteroidal Aromatase Inhibitors Identified through aMultidisciplinary Medicinal Chemistry Approach Synthesis and Monoamine Transporter Binding Properties of2,3-Diaryltropanes Drug Discovery Handbook Edited by Shayne CoxGad. Wiley-Interscience, Hoboken, NJ. 2005. xix + 1471pp. 16 × 24 cm. ISBN 0471213845. $160.00. Synthesis of Two 3,5-Disubstituted Sulfonamide Catechol Ligands andEvaluation of Their Iron(III) Complexes for Use as MRI Contrast Agents Structural, Mutagenic, and Kinetic Analysis of the Binding of Substrates andInhibitors of Human Phenylethanolamine N-Methyltransferase Statistical Tools for Virtual Screening SAR by MS: Discovery of a New Class ofRNA-Binding Small Molecules for theHepatitis C Virus: Internal RibosomeEntry Site IIA Subdomain Benzophenone-Based Farnesyltransferase Inhibitors with High Activity againstTrypanosoma cruzi Synthesis and Evaluation of Quindoline Derivatives as G-Quadruplex Inducingand Stabilizing Ligands and Potential Inhibitors of Telomerase Urotensin-II Receptor Ligands. From Agonist to Antagonist Activity Synthesis and Pharmacological Characterization ofexo-2-(2‘-Chloro-5-pyridinyl)-7-(endo and exo)-aminobicyclo[2.2.1]heptanes asNovel Epibatidine Analogues Specific Targeting Highly Conserved Residues in the HIV-1 ReverseTranscriptase Primer Grip Region. Design, Synthesis, and BiologicalEvaluation of Novel, Potent, and Broad Spectrum NNRTIs with AntiviralActivity In Vitro Anticancer Activities and Optical Imaging of Novel IntercalativeNon-Cisplatin Conjugates Some Insights into the Stereochemistry of Inhibition of Macrophage MigrationInhibitory Factor with 2-Fluoro-p-hydroxycinnamate and Its Analogues fromMolecular Dynamics Simulations Application of Validated QSAR Models of D1 Dopaminergic Antagonists forDatabase Mining Exploratory Chemistry toward the Identification of a New Class of MultidrugResistance Reverters Inspired by Pervilleine and Verapamil Models Piperazinobenzopyranones and Phenalkylaminobenzopyranones: PotentInhibitors of Breast Cancer Resistance Protein (ABCG2) Antitumor Polycyclic Acridines. 17. Synthesis and Pharmaceutical Profiles ofPentacyclic Acridinium Salts Designed To Destabilize Telomeric Integrity Random Chemistry as a New Tool for the Generation of Small CompoundLibraries: Development of a New Acetylcholinesterase Inhibitor Light-Induced Anticancer Activity of [RuCl2(DMSO)4] Complexes Tricyclic Pyrazoles. 3. Synthesis, Biological Evaluation, and MolecularModeling of Analogues of the Cannabinoid Antagonist8-Chloro-1-(2‘,4‘-dichlorophenyl)-N-piperidin-1-yl-1,4,5,6-tetrahydrobenzo[6,7]cyclohepta[1,2-c]pyrazole-3-carboxamide 1-Benzhydryl-3-phenylurea and 1-Benzhydryl-3-phenylthiourea Derivatives: New Templates among the CB1 Cannabinoid Receptor Inverse Agonists Analysis of Peptide−Protein Binding Using Amino Acid Descriptors: Predictionand Experimental Verification for Human Histocompatibility ComplexHLA-A*0201 Synthesis and Evaluation of Estrogen Receptor Ligands with BridgedOxabicyclic Cores Containing a Diarylethylene Motif: Estrogen Antagonists ofUnusual Structure Synthesis of N-{4-[(2,4-Diamino-5-methyl-4,7-dihydro-3H-pyrrolo[2,3-d]pyrimidin-6-yl)thio]benzoyl}-l-glutamic Acid andN-{4-[(2-Amino-4-oxo-5-methyl-4,7-dihydro-3H-pyrrolo[2,3-d]pyrimidin-6-yl)thio]benzoyl}-l-glutamic Acid as Dual Inhibitors of DihydrofolateReductase and Thymidylate Synthase and as Potential Antitumor Agents Radioiodinated Flavones for in Vivo Imaging of β-Amyloid Plaques in the Brain Annual Review of Biochemistry. Volume 74 Edited by Roger D. Kornberg, Christian R. H. Raetz, JamesE. Rothman, and Jeremy W. Thorner. Annual Reviews,Palo Alto, CA. 2005. x + 1010 pp. 15 × 25 cm. ISBN0-8243-0874-3. $88.00. Inhibitors of Tripeptidyl Peptidase II. 3. Derivation of Butabindide bySuccessive Structure Optimizations Leading to a Potential General Approach toDesigning Exopeptidase Inhibitors Irreversible Inactivation of Trypanothione Reductase by Unsaturated MannichBases: A Divinyl Ketone as Key Intermediate Virtual Screening of Novel CB2 Ligands Using a Comparative Model of theHuman Cannabinoid CB2 Receptor Cellular Apoptosis and Cytotoxicity of Phenolic Compounds: A QuantitativeStructure−Activity Relationship Study Anilinodialkoxyquinazolines: Screening Epidermal Growth Factor ReceptorTyrosine Kinase Inhibitors for Potential Tumor Imaging Probes Discovery of Novel and Potent Small-Molecule Inhibitors of NO and CytokineProduction as Antisepsis Agents: Synthesis and Biological Activity of Alkyl6-(N-Substituted sulfamoyl)cyclohex-1-ene-1-carboxylate Synthesis, Molecular Modeling Studies, and Selective Inhibitory Activityagainst Monoamine Oxidase of 1-Thiocarbamoyl-3,5-diaryl-4,5-dihydro-(1H)-pyrazole Derivatives Synthesis and Biological Activity of Anticancer Ether Lipids That AreSpecifically Released by Phospholipase A2 in Tumor Tissue Synthesis and 3D QSAR of New Pyrazolo[3,4-b]pyridines: Potent and SelectiveInhibitors of A1 Adenosine Receptors Identification of Borinic Esters as Inhibitors of Bacterial Cell Growth andBacterial Methyltransferases, CcrM and MenH Determinants of Corticotropin ReleasingFactor. Receptor Selectivity of Corticotropin ReleasingFactor Related Peptides. SAR and 3D-QSAR Studies on Thiadiazolidinone Derivatives: Exploration ofStructural Requirements for Glycogen Synthase Kinase 3 Inhibitors [N-Ethyl- and [N,N‘-Diethyl-1,2-bis(2,6-difluoro-3-hydroxyphenyl)-ethylenediamine]dichloroplatinum(II): Structure and Cytotoxic/EstrogenicActivity in Breast Cancer Cells Ligand Docking in the Gastric H+/K+-ATPase: Homology Modeling of ReversibleInhibitor Binding Sites Design, Synthesis, and Biological Evaluation of Dual Binding SiteAcetylcholinesterase Inhibitors: New Disease-Modifying Agents for Alzheimer'sDisease Structure−Activity Relationship of Triazafluorenone Derivatives as Potent andSelective mGluR1 Antagonists Damicoside from Axinella damicornis: The Influence of a GlycosylatedGalactose 4-OH Group on the Immunostimulatory Activity ofα-Galactoglycosphingolipids Synthesis and Characterization of theNovel Fluorescent Prolyl OligopeptidaseInhibitor 4-Fluoresceinthiocarbamoyl-6-aminocaproyl-l-prolyl-2(S)-(Hydroxy-acetyl)pyrrolidine Novel Tetralone-Derived Retinoic Acid Metabolism Blocking Agents: Synthesisand in Vitro Evaluation with Liver Microsomal and MCF-7 CYP26A1 Cell Assays Δ9-Tetrahydrocannabinol Immunochemical Studies: Haptens, MonoclonalAntibodies, and a Convenient Synthesis of RadiolabeledΔ9-Tetrahydrocannabinol Identification of Novel and ImprovedAntimitotic Agents Derived fromNoscapine 7-(1,1-Dimethylethyl)-6-(2-ethyl-2H-1,2,4-triazol-3-ylmethoxy)-3-(2-fluorophenyl)-1,2,4-triazolo[4,3-b]pyridazine: AFunctionally Selective γ-AminobutyricAcidA (GABAA) α2/α3-Subtype SelectiveAgonist That Exhibits Potent AnxiolyticActivity but Is Not Sedating in AnimalModels Frontiers in Natural Products Chemistry. Volume1 Edited by Atta-ur-Rahman, M. Iqbal Choudhary, andKhalid M. Khan. Bentham Science Publishers, Ltd.,Hilversum, The Netherlands. 2005. xiii + 234 pp. 16.5× 25 cm. ISBN 90-77527-044. $130.00.

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